BDBM595691 4-(3-(3-Fluoro-4-(4-methylpiperazin-1-yl)phenyl)-1H-pyrazolo[4,3-b]pyridin-5-yl)-3-isopropyl-1-methylpiperazin-2-one::US11591329, Ex. No. 18

SMILES CC(C)C1N(CCN(C)C1=O)c1ccc2[nH]nc(-c3ccc(N4CCN(C)CC4)c(F)c3)c2n1

InChI Key InChIKey=ICOYFUBCQGNVBP-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 595691   

TargetFibroblast growth factor receptor 3(Human)
Incyte

US Patent
LigandPNGBDBM595691(US11591329, Ex. No. 18 | 4-(3-(3-Fluoro-4-(4-methy...)
Affinity DataIC50: 10nMAssay Description:The inhibitor potency of the exemplified compounds was measured in an enzyme assay that measures peptide phosphorylation using FRET measurements to d...More data for this Ligand-Target Pair
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Date in BDB:
4/14/2023
Entry Details
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