BDBM595682 3-(Cyclopropylmethyl)-1-methyl-4-(3-(1-methyl-1H-pyrazol-4-yl)-1H-pyrazolo[4,3-b]pyridin-5-yl)piperazin-2-one::US11591329, Ex. No. 9

SMILES CN1CCN(C(CC2CC2)C1=O)c1ccc2[nH]nc(-c3cnn(C)c3)c2n1

InChI Key InChIKey=CRMRHFWRXXVBQT-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 595682   

TargetFibroblast growth factor receptor 3(Human)
Incyte

US Patent
LigandPNGBDBM595682(US11591329, Ex. No. 9 | 3-(Cyclopropylmethyl)-1-me...)
Affinity DataIC50: 20nMAssay Description:The inhibitor potency of the exemplified compounds was measured in an enzyme assay that measures peptide phosphorylation using FRET measurements to d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/14/2023
Entry Details
Go to US Patent