BDBM595677 3-Methyl-8-(3-(1-methyl-1H-pyrazol-4-yl)-1H-pyrazolo[4,3-b]pyridin-5-yl)-3,8-diazabicyclo[3.2.1]octan-2-one::US11591329, Ex. No. 4

SMILES CN1CC2CCC(N2c2ccc3[nH]nc(-c4cnn(C)c4)c3n2)C1=O

InChI Key InChIKey=IOKOTCFKNYVDJI-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 595677   

TargetFibroblast growth factor receptor 3(Human)
Incyte

US Patent
LigandPNGBDBM595677(US11591329, Ex. No. 4 | 3-Methyl-8-(3-(1-methyl-1H...)
Affinity DataIC50: 10nMAssay Description:The inhibitor potency of the exemplified compounds was measured in an enzyme assay that measures peptide phosphorylation using FRET measurements to d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/14/2023
Entry Details
Go to US Patent