BDBM590852 1-(4-fluorobenzyl)-6-(oxetan-3-yl)-2- oxo-N-(spiro[3.3]heptan-2-yl)-1,2- dihydro-1,8-naphthyridine-3-carboxamide::US11564928, Compound 102

SMILES Fc1ccc(Cn2c3ncc(cc3cc(C(=O)NC3CC4(CCC4)C3)c2=O)C2COC2)cc1

InChI Key InChIKey=LYSFLVJHFZQXDA-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 590852   

TargetCannabinoid receptor 2(Human)
Teon Therapeutics

US Patent
LigandPNGBDBM590852(US11564928, Compound 102 | 1-(4-fluorobenzyl)-6-(o...)
Affinity DataIC50: 2.30nMAssay Description:CB1R binding protocol involves the use of the same solution buffer used for both incubation and washing reaction (Tris-HCl, 50 mM; EDTA, 2.5 mM; MgCl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2023
Entry Details
Go to US Patent

TargetCannabinoid receptor 1(Human)
Teon Therapeutics

US Patent
LigandPNGBDBM590852(US11564928, Compound 102 | 1-(4-fluorobenzyl)-6-(o...)
Affinity DataIC50: 1.61E+3nMAssay Description:CB1R binding protocol involves the use of the same solution buffer used for both incubation and washing reaction (Tris-HCl, 50 mM; EDTA, 2.5 mM; MgCl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2023
Entry Details
Go to US Patent