BDBM590763 4-hydroxy-6-(4- methoxyphenyl)-1-(2- morpholinoethyl)-2-oxo-N- (spiro[3.3]heptan-2-yl)-1,2- dihydro-1,8-naphthyridine-3-carboxamide::US11564928, Compound 10

SMILES COc1ccc(cc1)-c1cnc2n(CCN3CCOCC3)c(=O)c(C(=O)NC3CC4(CCC4)C3)c(O)c2c1

InChI Key InChIKey=AYCFFHZZYFINHN-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 590763   

TargetCannabinoid receptor 2(Human)
Teon Therapeutics

US Patent
LigandPNGBDBM590763(US11564928, Compound 10 | 4-hydroxy-6-(4- methoxy...)
Affinity DataIC50: 7nMAssay Description:CB1R binding protocol involves the use of the same solution buffer used for both incubation and washing reaction (Tris-HCl, 50 mM; EDTA, 2.5 mM; MgCl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2023
Entry Details
Go to US Patent

TargetCannabinoid receptor 1(Human)
Teon Therapeutics

US Patent
LigandPNGBDBM590763(US11564928, Compound 10 | 4-hydroxy-6-(4- methoxy...)
Affinity DataIC50: 1.00E+4nMAssay Description:CB1R binding protocol involves the use of the same solution buffer used for both incubation and washing reaction (Tris-HCl, 50 mM; EDTA, 2.5 mM; MgCl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2023
Entry Details
Go to US Patent