BDBM573814 (1R,2S,5S)-8-(benzo [b]thiophene- 3-ylmethyl) (methyl)carbamoyl)-3- (diphenylcarbamoyl)- 3,8-diazabicyclo [3.2.1]octane- 2-carboxylic acid::US11453690, Example C246::US11453690, Example C279

SMILES CN(Cc1csc2ccccc12)C(=O)N1[C@H]2CC[C@@H]1[C@H](N(C2)C(=O)N(c1ccccc1)c1ccccc1)C(O)=O

InChI Key

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 573814   

TargetType-2 angiotensin II receptor(Human)
Beijing Tide Pharmaceutical

US Patent
LigandPNGBDBM573814(US11453690, Example C246 | (1R,2S,5S)-8-(benzo [b]...)
Affinity DataIC50: 10.1nMAssay Description:Measurement of Inhibitory Activity on AT1 Receptor (AT4R)/AT2 Receptor (AT2R)Through the following steps, the inhibitory activity of the compound on ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2022
Entry Details
Go to US Patent

TargetType-2 angiotensin II receptor(Human)
Beijing Tide Pharmaceutical

US Patent
LigandPNGBDBM573814(US11453690, Example C246 | (1R,2S,5S)-8-(benzo [b]...)
Affinity DataIC50: 24.2nMAssay Description:Measurement of Inhibitory Activity on AT1 Receptor (AT4R)/AT2 Receptor (AT2R)Through the following steps, the inhibitory activity of the compound on ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2022
Entry Details
Go to US Patent