BDBM573782 (1R,2S,5S)-8- (cyclopropyl(thiazole- 4-ylmethyl) carbamoyl)-3- (diphenylcarbamoyl)- 3,8-diazabicyclo [3.2.1]octane- 2-carboxylic acid::US11453690, Example C206

SMILES OC(=O)[C@@H]1[C@H]2CC[C@@H](CN1C(=O)N(c1ccccc1)c1ccccc1)N2C(=O)N(Cc1cscn1)C1CC1

InChI Key

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 573782   

TargetType-2 angiotensin II receptor(Human)
Beijing Tide Pharmaceutical

US Patent
LigandPNGBDBM573782(US11453690, Example C206 | (1R,2S,5S)-8- (cyclopro...)
Affinity DataIC50: 10.1nMAssay Description:Measurement of Inhibitory Activity on AT1 Receptor (AT4R)/AT2 Receptor (AT2R)Through the following steps, the inhibitory activity of the compound on ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2022
Entry Details
Go to US Patent