BDBM573774 (1R,2S,5S)-8- (cyclopropyl(5- methylthiophen-3- yl)methyl)carbamoyl)- 3- (diphenylcarbamoyl)- 3,8-diazabicyclo [3.2.1]octane- 2-carboxylic acid::US11453690, Example C197

SMILES Cc1cc(CN(C2CC2)C(=O)N2[C@H]3CC[C@@H]2[C@H](N(C3)C(=O)N(c2ccccc2)c2ccccc2)C(O)=O)cs1

InChI Key

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 573774   

TargetType-2 angiotensin II receptor(Human)
Beijing Tide Pharmaceutical

US Patent
LigandPNGBDBM573774(US11453690, Example C197 | (1R,2S,5S)-8- (cyclopro...)
Affinity DataIC50: 5.52nMAssay Description:Measurement of Inhibitory Activity on AT1 Receptor (AT4R)/AT2 Receptor (AT2R)Through the following steps, the inhibitory activity of the compound on ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2022
Entry Details
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