BDBM573770 (1R,2S,5S)-3-(2,2- diphenylacetyl)-8- (ethyl(thiophene-3- ylmethyl) carbamoyl)-3,8- diazabicyclo [3.2.1]octane- 2-carboxylic acid::US11453690, Example C188

SMILES CCN(Cc1ccsc1)C(=O)N1[C@H]2CC[C@@H]1[C@H](N(C2)C(=O)C(c1ccccc1)c1ccccc1)C(O)=O

InChI Key

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 573770   

TargetType-2 angiotensin II receptor(Human)
Beijing Tide Pharmaceutical

US Patent
LigandPNGBDBM573770(US11453690, Example C188 | (1R,2S,5S)-3-(2,2- diph...)
Affinity DataIC50: 7.11nMAssay Description:Measurement of Inhibitory Activity on AT1 Receptor (AT4R)/AT2 Receptor (AT2R)Through the following steps, the inhibitory activity of the compound on ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2022
Entry Details
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