BDBM565698 US11407768, Compound MK-8722

SMILES O[C@@H]1CO[C@@H]2[C@@H](CO[C@H]12)Oc1nc2c(Cl)c(cnc2[nH]1)-c1ccc(cc1)-c1ccccc1

InChI Key InChIKey=VEGCGBKTFKSLJB-UHFFFAOYSA-N

Data  1 EC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 565698   

Target5'-AMP-activated protein kinase catalytic subunit alpha-1/subunit beta-1/subunit gamma-1(Human)
Kallyope

US Patent

LigandBDBM565698(US11407768, Compound MK-8722)Copy SMILESCopy InChI

Affinity DataEC50:  10.4nMAssay Description:Compound effect on AMPK enzyme activation was determined in a cell-free format with a 12-point concentration curve. The ADP-Glo detection system was ...More data for this Ligand-Target Pair

Target InfoPDB
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sidSimilars

In Depth
Date in BDB:
11/5/2022
Entry Details
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