BDBM559569 US11370795, Compound (P1)::US11608342, Compound (P1)::US20250019381, Compound (P1)

SMILES Fc1ccc(cc1)-c1ncc2n1cc(CN1CC(C1)Oc1ccncc1)[nH]c2=O

InChI Key InChIKey=OPPJESMUQLKXLM-UHFFFAOYSA-N

Data  6 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 6 hits for monomerid = 559569   

LigandPNGBDBM559569(US11608342, Compound (P1) | US11370795, Compound (...)
Affinity DataIC50: 42nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/25/2022
Entry Details
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LigandPNGBDBM559569(US11608342, Compound (P1) | US11370795, Compound (...)
Affinity DataIC50: 4.51E+4nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/25/2022
Entry Details
Go to US Patent

LigandPNGBDBM559569(US11608342, Compound (P1) | US11370795, Compound (...)
Affinity DataIC50: 42nMAssay Description:A PDE9 assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/5/2023
Entry Details
Go to US Patent

LigandPNGBDBM559569(US11608342, Compound (P1) | US11370795, Compound (...)
Affinity DataIC50: 4.51E+4nMAssay Description:PDE1 assays were performed as follows: the assays was performed in 60 μL samples containing a fixed amount of the PDE1 enzym1 (sufficient to con...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/5/2023
Entry Details
Go to US Patent

LigandPNGBDBM559569(US11608342, Compound (P1) | US11370795, Compound (...)
Affinity DataIC50: 42nMAssay Description:Non-limiting examples of PDE9 inhibitors of formula (II) are disclosed in WO 2013/110768, the contents of which are incorporated herein by reference ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2025
Entry Details
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LigandPNGBDBM559569(US11608342, Compound (P1) | US11370795, Compound (...)
Affinity DataIC50: 4.51E+4nMAssay Description:Non-limiting examples of PDE9 inhibitors of formula (II) are disclosed in WO 2013/110768, the contents of which are incorporated herein by reference ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2025
Entry Details
Go to US Patent