BDBM551244 7-Fluoro-5-(2-isopropyl-6-methyl-pyrrolo[2,3-b]pyridin-1-yl)indolin-2-one;::US11312712, Example 362

SMILES CC(C)c1cc2ccc(C)nc2n1-c1cc2CC(=O)Nc2c(F)c1

InChI Key InChIKey=LYYJJOICYBLSJE-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 551244   

TargetVoltage-dependent calcium channel gamma-8 subunit(Human)
Janssen Pharmaceutica

US Patent
LigandPNGBDBM551244(US11312712, Example 362 | 7-Fluoro-5-(2-isopropyl-...)
Affinity DataIC50: 0.0400nMAssay Description:An in vitro assay was used to determine the potency of test compounds as inhibitors of the glutamate response of the channel formed by GluA1o-γ8...More data for this Ligand-Target Pair
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Date in BDB:
8/6/2022
Entry Details
US Patent