BDBM537043 US11897851, Compound 143

SMILES CCn1cncc1Cn1c(CCC(O)=O)cnc1CN1CCC(CC1)c1cccc2OC(C)(Oc12)c1ccc(Cl)cc1F

InChI Key InChIKey=JDGVMZRHJITZQD-UHFFFAOYSA-N

Data  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 537043   

TargetGlucagon-like peptide 1 receptor(Human)
Gasherbrum Bio

US Patent
LigandPNGBDBM537043(US11897851, Compound 143)
Affinity DataEC50:  0.00600nMAssay Description:To optimize functional activity directed toward Gas coupling, a HEK293/CRE-Luc cell line developed by HDB stably expressing the GLP-1 Receptor was us...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2024
Entry Details
Go to US Patent