BDBM537016 (E)-3-(6-((4-(6-((4-chloro-2-fluorobenzyl)oxy)pyridin-2-yl)piperidin-1-yl)methyl)-5-((tetrahydrofuran-2-yl)methyl)pyridin-3-yl)acrylic acid ::US11897851, Compound 128

SMILES OC(=O)\C=C\c1cnc(CN2CCC(CC2)c2cccc(OCc3ccc(Cl)cc3F)n2)c(CC2CCCO2)c1

InChI Key InChIKey=DJEYHRJZVUVMAH-UHFFFAOYSA-N

Data  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 537016   

TargetGlucagon-like peptide 1 receptor(Human)
Gasherbrum Bio

US Patent
LigandPNGBDBM537016((E)-3-(6-((4-(6-((4-chloro-2-fluorobenzyl)oxy)pyri...)
Affinity DataEC50:  48.9nMAssay Description:To optimize functional activity directed toward Gas coupling, a HEK293/CRE-Luc cell line developed by HDB stably expressing the GLP-1 Receptor was us...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2024
Entry Details
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