BDBM536997 2-{2-[(4-{6-[(4-chloro-2-fluorophenyl)methoxy]pyridin-2-yl}piperidin-1-yl)methyl]-1-{[(2S)-oxetan-2-yl]methyl}-1H-imidazol-5-yl}cyclopropane-1-carboxylic acid ::US11897851, Compound 114a

SMILES Fc1cc(Cl)ccc1COc1cccc(n1)C1CCN(Cc2ncc(C3CC3)n2C[C@@H]2CCO2)CC1

InChI Key InChIKey=MLQYCENXYUTNAS-UHFFFAOYSA-N

Data  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 536997   

TargetGlucagon-like peptide 1 receptor(Human)
Gasherbrum Bio

US Patent
LigandPNGBDBM536997(2-{2-[(4-{6-[(4-chloro-2-fluorophenyl)methoxy]pyri...)
Affinity DataEC50:  9.40nMAssay Description:To optimize functional activity directed toward Gas coupling, a HEK293/CRE-Luc cell line developed by HDB stably expressing the GLP-1 Receptor was us...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2024
Entry Details
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