BDBM536987 (S,E)-3-(2-((4-(6-((4-chloro-2-fluorobenzyl)oxy)pyridin-2-yl)piperidin-1-yl)methyl)-1-(oxetan-2-ylmethyl)-1H-imidazol-5-yl)acrylic acid ::US11897851, Compound 103a

SMILES Fc1cc(Cl)ccc1COc1cccc(n1)C1CCN(Cc2ncc(C=C)n2C[C@@H]2CCO2)CC1

InChI Key InChIKey=XQQGSZHFGIAHRC-UHFFFAOYSA-N

Data  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 536987   

TargetGlucagon-like peptide 1 receptor(Human)
Gasherbrum Bio

US Patent
LigandPNGBDBM536987((S,E)-3-(2-((4-(6-((4-chloro-2-fluorobenzyl)oxy)py...)
Affinity DataEC50:  0.0930nMAssay Description:To optimize functional activity directed toward Gas coupling, a HEK293/CRE-Luc cell line developed by HDB stably expressing the GLP-1 Receptor was us...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2024
Entry Details
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