BDBM534177 6-Cyclopropyl-N-[(2-methyl-8-quinolyl)sulfonyl]-4-(trifluoromethyl)benzofuran-2-carboxamide::WO2022081842, Example 50

SMILES Cc1ccc2cccc(c2n1)S(=O)(=O)NC(=O)c1cc2c(cc(cc2o1)C1CC1)C(F)(F)F

InChI Key InChIKey=XGZWWVOYBHRFHY-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 534177   

TargetHistone acetyltransferase KAT6A [507-778](Human)
The Broad Institute

WIPO
LigandPNGBDBM534177(WO2022081842, Example 50 | 6-Cyclopropyl-N-[(2-met...)
Affinity DataIC50: 5.55nMAssay Description: Kat6a inhibitory activities of the compounds described in the present invention were quantified using a Fluorescence Resonance Energy Transfer (TR-F...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2022
Entry Details
WIPO WO2022081842