BDBM534024 6-(Azetidin-1-yl)-N-[2-(cyclopropyloxy)benzene-1-sulfonyl]-4-fluoro-1-benzofuran- 2-carboxamide::WO2022081807, Example 131

SMILES Fc1cc(cc2oc(cc12)C(=O)NS(=O)(=O)c1ccccc1OC1CC1)N1CCC1

InChI Key InChIKey=JIDSZOUWGCYNTO-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 534024   

TargetHistone acetyltransferase KAT6A [507-778](Human)
The Broad Institute

WIPO
LigandPNGBDBM534024(WO2022081807, Example 131 | 6-(Azetidin-1-yl)-N-[2...)
Affinity DataIC50: 23nMAssay Description:Kat6a inhibitory activities of the compounds described in the present invention were quantified using a Fluorescence Resonance Energy Transfer (TR-FR...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2022
Entry Details
WIPO WO2022081807

TargetHistone acetyltransferase KAT6B(Human)
The Broad Institute

WIPO
LigandPNGBDBM534024(WO2022081807, Example 131 | 6-(Azetidin-1-yl)-N-[2...)
Affinity DataIC50: 23nMAssay Description:Kat6b inhibitory activities of the compounds described in the present invention were quantified using a Fluorescence Resonance Energy Transfer (TR-FR...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2022
Entry Details
WIPO WO2022081807