BDBM533902 6-(Azetidin-1-yl)-N-([1,T-biphenyl]-2-sulfonyl)-1-benzofuran-2-carboxamide::WO2022081807, Example 26

SMILES O=C(NS(=O)(=O)c1ccccc1-c1ccccc1)c1cc2ccc(cc2o1)N1CCC1

InChI Key InChIKey=HDFSCNSLBMMCMW-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 533902   

TargetHistone acetyltransferase KAT6A [507-778](Human)
The Broad Institute

WIPO
LigandPNGBDBM533902(WO2022081807, Example 26 | 6-(Azetidin-1-yl)-N-([1...)
Affinity DataIC50: 145nMAssay Description:Kat6a inhibitory activities of the compounds described in the present invention were quantified using a Fluorescence Resonance Energy Transfer (TR-FR...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2022
Entry Details
WIPO WO2022081807

TargetHistone acetyltransferase KAT6B(Human)
The Broad Institute

WIPO
LigandPNGBDBM533902(WO2022081807, Example 26 | 6-(Azetidin-1-yl)-N-([1...)
Affinity DataIC50: 292nMAssay Description:Kat6b inhibitory activities of the compounds described in the present invention were quantified using a Fluorescence Resonance Energy Transfer (TR-FR...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/24/2022
Entry Details
WIPO WO2022081807