BDBM528489 5-(1H-Indazol-5-yl)-2-(pyridin-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidin-7(4H)-one::US11191765, Example 3

SMILES O=c1cc([nH]c2nc(nn12)-c1ccccn1)-c1ccc2[nH]ncc2c1

InChI Key InChIKey=KRHXODCCUZVENL-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 528489   

TargetPAS domain-containing serine/threonine-protein kinase(Human)
Bioenergenix

US Patent

LigandBDBM528489(US11191765, Example 3 | 5-(1H-Indazol-5-yl)-2-(pyr...)Copy SMILESCopy InChI

Affinity DataIC50: 1.00E+4nMAssay Description:The aim of the FRET assay is to determine the inhibition potential of test compounds on targeted kinase. This assay platform provides a homogenous sc...More data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
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Ligand InfoPC cidPC sidSimilars

In Depth
Date in BDB:
4/17/2022
Entry Details
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