BDBM524304 Preparation of 4'-(4-methyl-1-((2-(piperidin-1-yl)thiazol-4-yl)methyl)-1H-pyrrole-2-carboxamido)-[1,1'-biphenyl]-4-carboxylic Acid::US11168080, Compound A-71

SMILES Cc1cc(C(=O)Nc2ccc(cc2)-c2ccc(cc2)C(O)=O)n(Cc2csc(n2)N2CCCCC2)c1

InChI Key InChIKey=KSGQTRGOZMODMQ-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 524304   

TargetDynamin-1-like protein(Human)
Mitobridge

US Patent
LigandPNGBDBM524304(Preparation of 4'-(4-methyl-1-((2-(piperidin-1-yl)...)
Affinity DataIC50: 720nMAssay Description:The GTPase activity of Drp1 was assayed using a colorimetric assay similar to as described previously by Leonard M. et al. Robust colorimetric assays...More data for this Ligand-Target Pair
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Date in BDB:
3/27/2022
Entry Details
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