BDBM506987 4-hydroxy-2-(2-hydroxyphenyl)-N- methoxy-N-methyl-1,3-thiazole-5- carboxamide::US11046662, Compound 12

SMILES CON(C)C(=O)c1sc(nc1O)-c1ccccc1O

InChI Key InChIKey=UFNWXHVCAXKDMI-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 506987   

LigandPNGBDBM506987(4-hydroxy-2-(2-hydroxyphenyl)-N- methoxy-N-methyl-...)
In Depth
Date in BDB:
12/27/2021
Entry Details
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LigandPNGBDBM506987(4-hydroxy-2-(2-hydroxyphenyl)-N- methoxy-N-methyl-...)
Affinity DataIC50: 66nMAssay Description:Inhibition of human TRPM8 expressed in HEK293 cells assessed as reduction in ethyl 4-methoxy-2-phenylthiazole-5-carboxylate induced Ca2+ efflux prein...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed