BDBM50668042 CHEMBL6188778

SMILES Cc1ccc(S(=O)(=O)c2c[nH]c(SCC(=O)Nc3ccc(C(F)(F)F)cc3)nc2=O)cc1Cl

InChI Key InChIKey=LCVRBHCJJZWVHH-UHFFFAOYSA-N

Data  1 KI  1 IC50  4 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 6 hits for monomerid = 50668042   

TargetChemerin-like receptor 2(Homo sapiens)
Leipzig University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50668042BDBM50668042(CHEMBL6188778)
Affinity DataEC50:  7nMAssay Description:Antagonist activity at eYFP-tagged human GPR1 transfected in HEK293 cells assessed as inhibition of TAMRA-labeled-(RG4)-C9 induced receptor internali...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetChemerin-like receptor 1(Human)
Leipzig University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50668042BDBM50668042(CHEMBL6188778)
Affinity DataEC50:  10nMAssay Description:Antagonist activity at eYFP-tagged human CMKLR1b transfected in C9-stimulated HEK293 cells co-transfected with Galpha-delta6qi4myr assessed as inhibi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetChemerin-like receptor 1(Human)
Leipzig University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50668042BDBM50668042(CHEMBL6188778)
Affinity DataEC50:  47nMAssay Description:Antagonist activity at eYFP-tagged human CMKLR1b transfected in C9-stimulated HEK293 cells co-transfected with Galpha-delta6qi4myr assessed as inhibi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetChemerin-like receptor 1(Human)
Leipzig University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50668042BDBM50668042(CHEMBL6188778)
Affinity DataEC50:  202nMAssay Description:Antagonist activity at eYFP-tagged human CMKLR1b transfected in HEK293 cells co-transfected with Galpha-delta6qi4myr assessed as inhibition of TAMRA-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetChemerin-like receptor 2(Homo sapiens)
Leipzig University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50668042BDBM50668042(CHEMBL6188778)
Affinity DataKi:  1.48E+3nMAssay Description:Displacement of TAMRA-labeled chemerin 9 from Nluc-tagged GPR1 (unknown origin) transfected in HEK293 cells assessed as inhibition constant incubated...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetChemerin-like receptor 1(Human)
Leipzig University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50668042BDBM50668042(CHEMBL6188778)
Affinity DataIC50: 3.70E+4nMAssay Description:Antagonist activity at eYFP-tagged human CMKLR1b transfected in C9-stimulated HEK293 cells co-transfected with Galpha-delta6qi4myr assessed as inhibi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed