BDBM50629987 CHEMBL5417465
SMILES ClC(Cl)C(=O)NCCCCC(=O)Nc1ccc(cc1)[As]1SCCCS1
InChI Key InChIKey=VUZLJKJFKWPURT-UHFFFAOYSA-N
Data 1 EC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 50629987
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial(Human)
Wuhan University
Curated by ChEMBL
Wuhan University
Curated by ChEMBL
Affinity DataEC50: 930nMAssay Description:Inhibition of PDK1 (unknown origin) incubated for 30 mins in presence of ATP by kinase glo luminescent kinase assayMore data for this Ligand-Target Pair