BDBM50623720 CHEMBL5430692

SMILES COc1cc(CN(c2ccc(I)cc2F)c2c(F)c(F)ccc2C(=O)NOC[C@H](O)CO)c(cc1OC)[N+]([O-])=O

InChI Key InChIKey=IZHGONBICPNYMQ-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50623720   

TargetDual specificity mitogen-activated protein kinase kinase 1(Human)
Peking University

Curated by ChEMBL

LigandBDBM50623720(CHEMBL5430692)Copy SMILESCopy InChI

Affinity DataIC50: 878nMAssay Description:Inhibition of MEK1 (unknown origin) incubated for 1 hrs in the presence of ATP by FRET-based Z'-Lyte assayMore data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoSimilars

In Depth
Date in BDB:
12/17/2024
Entry Details
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