BDBM50623319 CHEMBL5423651

SMILES CC(C)Nc1nc2ccc(cc2n1C1CCN(CC1)c1ccc(cc1)C(C)(C)C#N)C#N

InChI Key InChIKey=UYFLPAHZXSVYSO-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50623319   

TargetTransient receptor potential cation channel subfamily V member 4(Human)
Beijing Institute of Pharmacology and Toxicology

Curated by ChEMBL
LigandPNGBDBM50623319(CHEMBL5423651)
Affinity DataIC50: 79nMAssay Description:Antagonist activity at TRPV4 (unknown origin) expressed in Flp-In-CHO cells assessed as inhibition of GSK1016790A induced Ca2+ influx by calcium imag...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed