BDBM50617207 CHEMBL5400532

SMILES Cc1nnc2CN[C@@H](c3c4C[C@H](Cc4sc3-n12)C(=O)NC1CCC(F)(F)CC1)c1ccccc1Cl

InChI Key InChIKey=BUPZLUDNAYIQNE-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50617207   

TargetPlatelet-activating factor receptor(Human)
Smith, Gambrell & Russell

Curated by ChEMBL
LigandPNGBDBM50617207(CHEMBL5400532)
Affinity DataIC50: 1.30nMAssay Description:Antagonist activity at human PAFR expressed in HEK293 cells assessed as inhibition of PAF C-16 ligand induced receptor activation preincubated for 90...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed