BDBM50608078 CHEMBL1876546

SMILES Cc1cc(C)c2CCCNc2n1

InChI Key InChIKey=DXIRHDQUVVQLGI-UHFFFAOYSA-N

Data  3 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50608078   

TargetE3 ubiquitin-protein ligase UHRF1(Human)
University of S£O Paulo

Curated by ChEMBL
LigandPNGBDBM50608078(CHEMBL1876546)
Affinity DataEC50:  4.50E+4nMAssay Description:Inhibition of His tagged UHRF1 tandem Tudor domain (unknown origin) using biotinylated-H3K9me3 peptide as substrate incubated for 1 hr by TR-FRET ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetE3 ubiquitin-protein ligase UHRF1(Human)
University of S£O Paulo

Curated by ChEMBL
LigandPNGBDBM50608078(CHEMBL1876546)
Affinity DataEC50:  4.51E+4nMAssay Description:Inhibition of UHRF1 (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetE3 ubiquitin-protein ligase UHRF1(Human)
University of S£O Paulo

Curated by ChEMBL
LigandPNGBDBM50608078(CHEMBL1876546)
Affinity DataEC50:  5.67E+4nMAssay Description:Inhibition of UHRF1 (unknown origin) by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed