BDBM50601673 CHEMBL5206379

SMILES CCCCCCCCCCCOc1cccc(CCC(=O)NC[C@@H](O)COP(O)(=O)OC[C@H](NC(=O)c2ccc(C)cc2)C(O)=O)c1

InChI Key InChIKey=KLIGFZBOUZXBPW-UHFFFAOYSA-N

Data  2 IC50  2 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50601673   

TargetProbable G-protein coupled receptor 174(Mouse)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50601673(CHEMBL5206379)
Affinity DataEC50:  9nMAssay Description:Partial agonist activity at mouse GPR174 transfected in human HEK293FT cells co-transfected with AP-TGFalpha assessed as AP-TGFalpha release incubate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetProbable G-protein coupled receptor 174(Mouse)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50601673(CHEMBL5206379)
Affinity DataEC50:  9.5nMAssay Description:Partial agonist activity at mouse GPR174 transfected in human HEK293FT cells co-transfected with AP-TGFalpha assessed as AP-TGFalpha release incubate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetProbable G-protein coupled receptor 174(Mouse)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50601673(CHEMBL5206379)
Affinity DataIC50: 190nMAssay Description:Antagonist activity at mouse GPR174 transfected in human HEK293FT cells co-transfected with AP-TGFalpha assessed as inhibition of LysoPalloT-NH-C3-ph...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetProbable G-protein coupled receptor 174(Mouse)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50601673(CHEMBL5206379)
Affinity DataIC50: 186nMAssay Description:Antagonist activity at mouse GPR174 transfected in human HEK293FT cells co-transfected with AP-TGFalpha assessed as inhibition of LysoPalloT-NH-C3-ph...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed