BDBM50599842 CHEMBL5187587

SMILES Cc1nc2CN(CCc2c(Oc2ccc(F)cc2C(F)(F)F)n1)C1=C(Cl)C(=O)NC1=O

InChI Key InChIKey=DPATUHNUTTZBBN-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50599842   

TargetShort transient receptor potential channel 5(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50599842(CHEMBL5187587)
Affinity DataIC50: 125nMAssay Description:Inhibition of TRPC5 channel (unknown origin) expressed in HEK293 cells assessed as inhibition of EA-evoked Ca2+ entry by measuring reduction in intra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed