BDBM50582815 CHEMBL5078594

SMILES Cc1nn(C)cc1N1CCC(NC(=O)Nc2ccc(Br)cc2)C1=O

InChI Key InChIKey=WPOPBEUSMAIIMY-UHFFFAOYSA-N

Data  3 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50582815   

TargetN-formyl peptide receptor 2(Human)
Queen Mary University of London

Curated by ChEMBL
LigandPNGBDBM50582815(CHEMBL5078594)
Affinity DataEC50:  142nMAssay Description:Agonist activity at FPRL1 (unknown origin) expressed in CHO-K1 cells assessed as increase in calcium mobilization incubated for 2.5 hrs by cellular b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetN-formyl peptide receptor 2(Human)
Queen Mary University of London

Curated by ChEMBL
LigandPNGBDBM50582815(CHEMBL5078594)
Affinity DataEC50:  740nMAssay Description:Agonist activity at FPRL1 (unknown origin) expressed in CHO-K1 cells assessed as stimulation of beta-arrestin recruitment incubated for 150 mins by b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed
TargetN-formyl peptide receptor 2(Human)
Queen Mary University of London

Curated by ChEMBL
LigandPNGBDBM50582815(CHEMBL5078594)
Affinity DataEC50:  4.88E+3nMAssay Description:Agonist activity at human FPR2 expressed in HEK293-A cells assessed as ERK phosphorylation level incubated for 5 mins by ELISA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2023
Entry Details Article
PubMed