BDBM50579801 CHEMBL5088992

SMILES COC1=C(Cc2ccc(s2)-c2cn(Cc3ccccc3)cc(C(O)=O)c2=O)C(=O)N(C1)c1ccc2ccccc2c1

InChI Key InChIKey=YIGVZXFIAKXNEU-UHFFFAOYSA-N

Data  7 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 7 hits for monomerid = 50579801   

TargetHistone acetyltransferase p300(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50579801(CHEMBL5088992)
Affinity DataIC50: 4.90E+3nMAssay Description:Inhibition of EP300 (unknown origin) by AlphaLISA immunodetection assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetCREB-binding protein(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50579801(CHEMBL5088992)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of CBP (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetHistone acetyltransferase KAT7(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50579801(CHEMBL5088992)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of MYST2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetHistone acetyltransferase KAT6B(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50579801(CHEMBL5088992)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of MYST4 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetHistone acetyltransferase KAT2B(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50579801(CHEMBL5088992)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of PCAF (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetHistone acetyltransferase KAT2A(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50579801(CHEMBL5088992)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of GCN5 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetHistone acetyltransferase KAT5(Human)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50579801(CHEMBL5088992)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of TIP60 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed