BDBM50572972 CHEMBL4863245

SMILES Clc1cnn(CC(=O)Nc2cccc(c2)S(=O)(=O)NCCc2ccccn2)c(=O)c1Cl

InChI Key InChIKey=BVERKJPMUVLOFJ-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50572972   

TargetMethylosome protein 50/Protein arginine N-methyltransferase 5(Human)
The Broad Institute of Mit and Harvard

Curated by ChEMBL
LigandPNGBDBM50572972(CHEMBL4863245)
Affinity DataIC50: 1.92E+4nMAssay Description:Displacement of fluorophore-labeled RIOK1 from human PRMT5/WDR77 hetero octameric complex expressed in Sf9 cells by competition fluorescence polariza...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed