BDBM50572966 CHEMBL4849760

SMILES CN1CCN(CC1)S(=O)(=O)c1cc(NC(=O)Cn2ncc(Cl)c(Cl)c2=O)ccc1C

InChI Key InChIKey=PTMARBOXAAIGND-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50572966   

TargetMethylosome protein 50/Protein arginine N-methyltransferase 5(Human)
The Broad Institute of Mit and Harvard

Curated by ChEMBL
LigandPNGBDBM50572966(CHEMBL4849760)
Affinity DataIC50: 1.01E+4nMAssay Description:Displacement of fluorophore-labeled RIOK1 from human PRMT5/WDR77 hetero octameric complex expressed in Sf9 cells by competition fluorescence polariza...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed