BDBM50571944 CHEMBL4856749

SMILES CC(C)n1cc(C(=O)Nc2ccc(Oc3ncnc4CN(CCc34)C3CCN(C)CC3)c(F)c2)c(=O)n(-c2ccc(F)cc2)c1=O

InChI Key InChIKey=RYQKZEFCGLDZCP-UHFFFAOYSA-N

Data  4 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50571944   

TargetTyrosine-protein kinase receptor UFO(Human)
Eisai

Curated by ChEMBL
LigandPNGBDBM50571944(CHEMBL4856749)
Affinity DataIC50: 5.60nMAssay Description:Inhibition of Axl (unknown origin) by cell free assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2022
Entry Details Article
PubMed
TargetTyrosine-protein kinase Mer(Human)
Eisai

Curated by ChEMBL
LigandPNGBDBM50571944(CHEMBL4856749)
Affinity DataIC50: 31nMAssay Description:Inhibition of Mer (unknown origin) by cell free assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2022
Entry Details Article
PubMed
TargetTyrosine-protein kinase receptor UFO(Mouse)
Eisai

Curated by ChEMBL
LigandPNGBDBM50571944(CHEMBL4856749)
Affinity DataIC50: 13nMAssay Description:Inhibition of Axl in mouse BaF3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2022
Entry Details Article
PubMed
TargetTyrosine-protein kinase Mer(Mouse)
Eisai

Curated by ChEMBL
LigandPNGBDBM50571944(CHEMBL4856749)
Affinity DataIC50: 55nMAssay Description:Inhibition of Mer in mouse BaF3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2022
Entry Details Article
PubMed