BDBM50567334 CHEMBL4869045

SMILES FC(F)(F)c1ccc(NC(=O)c2ccn(Cn3cc(NC(=O)Cc4ccccc4)cn3)n2)cc1

InChI Key InChIKey=ATKARCDMBQCOAE-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50567334   

TargetHypoxia-inducible factor 1-alpha(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50567334(CHEMBL4869045)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of hypoxia-induced HIF1 alpha transcriptional activity in human HeLa cells transfected with luciferase reporter containing of HRE assessed...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed