BDBM50566795 CHEMBL4873003

SMILES COc1cc(OC)c(F)c(N2Cc3cnc4NC(=O)C5(CCN(C)CC5)c4c3N(C)C2=O)c1F

InChI Key InChIKey=DKYAEOVZIXOJNP-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50566795   

TargetFibroblast growth factor receptor 1(Human)
Incyte

Curated by ChEMBL
LigandPNGBDBM50566795(CHEMBL4873003)
Affinity DataIC50: 21nMAssay Description:Inhibition of human FGFR1 using biotinylated-EQEDEPEGDYFEWLE peptide as substrate incubated for 1 hr in presence of ATP by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed