BDBM50559211 CHEMBL4756631

SMILES Fc1ccc(CNC(=O)Cc2nnc(o2)-c2ccccn2)c(Cl)c1

InChI Key InChIKey=WOHXMCKHYRZMJE-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50559211   

TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Human)
Zhejiang University

Curated by ChEMBL

LigandBDBM50559211(CHEMBL4756631)Copy SMILESCopy InChI

Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of PI3Kalpha (unknown origin) using PIP2 as substrate measured after 1 hr by ADP-glo plus luminescence assayMore data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sidSimilars

In Depth
Date in BDB:
3/27/2022
Entry Details Article
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