BDBM50555224 CHEMBL4790482

SMILES Nc1nc(Cl)nc2n(Cc3cccc(n3)C3CCCC3)cnc12

InChI Key InChIKey=OJCLSOHWOVKXMM-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50555224   

TargetHigh affinity cAMP-specific and IBMX-insensitive 3',5'-cyclic phosphodiesterase 8A(Human)
Sun Yat-Sen University

Curated by ChEMBL

LigandBDBM50555224(CHEMBL4790482)Copy SMILESCopy InChI

Affinity DataIC50: 46nMAssay Description:Inhibition of PDE8A1 (480 to 820 residues) (unknown origin) expressed in Escherichia coli BL21 using [3H]-cAMP substrate incubated for 15 mins by liq...More data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sidSimilars

In Depth
Date in BDB:
3/25/2022
Entry Details Article
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