BDBM50554974 CHEMBL4777668

SMILES N[C@@H](CCNS(=O)(=O)c1ccc(Cl)cc1Cl)COc1cc(ccc1Cl)C#N

InChI Key InChIKey=NIPFFUIZKMPZRZ-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50554974   

TargetTransient receptor potential cation channel subfamily V member 4(Human)
Glaxosmithkline

Curated by ChEMBL

LigandBDBM50554974(CHEMBL4777668)Copy SMILESCopy InChI

Affinity DataIC50: 58nMAssay Description:Antagonist activity at human TRPV4 expressed in BHK or HEK MSR2 cells assessed as inhibition of TRPV4 agonist GSK634775 (EC80)-induced response incub...More data for this Ligand-Target Pair

Target InfoPDB
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sidSimilars

In Depth
Date in BDB:
3/25/2022
Entry Details Article
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