BDBM50554267 CHEMBL4760734

SMILES Fc1ccc(CNC(=O)c2cccc(Cn3cnc4ccc(cc4c3=O)-c3cn[nH]c3)c2)cc1

InChI Key InChIKey=WCMFMVGWKLJPNE-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50554267   

TargetBeta-adrenergic receptor kinase 1(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50554267(CHEMBL4760734)
Affinity DataIC50: 10nMAssay Description:Inhibition of human GRK2 by transcreener assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed