BDBM50548384 CHEMBL4762439
SMILES CCCCCc1cc(O)c([C@@H]2C=C(C)CC[C@H]2C(C)=C)c(O)c1Cc1c(CCCCC)cc(O)c([C@@H]2C=C(C)CC[C@H]2C(C)=C)c1O
InChI Key InChIKey=UMJIRNQSAUOZKO-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 10 hits for monomerid = 50548384
TargetTransient receptor potential cation channel subfamily M member 8(Rat)
University of Naples Federico Ii
Curated by ChEMBL
University of Naples Federico Ii
Curated by ChEMBL
Affinity DataIC50: 3.90E+3nMAssay Description:Antagonist activity at rat TRPM8 expressed in HEK293 cells assessed as inhibition of icilin-induced Ca2+ response preincubated for 5 mins followed by...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily A member 1(Rat)
University of Naples Federico Ii
Curated by ChEMBL
University of Naples Federico Ii
Curated by ChEMBL
Affinity DataIC50: 4.90E+3nMAssay Description:Antagonist activity at rat TRPA1 expressed in HEK293 cells assessed as inhibition of allylisothiocyanate-induced Ca2+ response preincubated for 5 min...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily A member 1(Rat)
University of Naples Federico Ii
Curated by ChEMBL
University of Naples Federico Ii
Curated by ChEMBL
Affinity DataEC50: 3.00E+3nMAssay Description:Agonist activity at rat TRPA1 stably transfected in HEK293 cells assessed as increase in calcium influx in presence of allylisothiocyanate by Fluo-4-...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 4(Rat)
University of Naples Federico Ii
Curated by ChEMBL
University of Naples Federico Ii
Curated by ChEMBL
Affinity DataIC50: 2.00E+4nMAssay Description:Antagonist activity at rat TRPV4 expressed in HEK293 cells assessed as inhibition of GSK1016790A-induced Ca2+ response preincubated for 5 mins follow...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 4(Rat)
University of Naples Federico Ii
Curated by ChEMBL
University of Naples Federico Ii
Curated by ChEMBL
Affinity DataEC50: 6.20E+3nMAssay Description:Agonist activity at rat TRPV4 stably transfected in HEK293 cells assessed as increase in calcium influx in presence of ionomycin by Fluo-4-AM dye bas...More data for this Ligand-Target Pair
Affinity DataIC50: 1.18E+4nMAssay Description:Antagonist activity at rat TRPV3 expressed in HEK293 cells assessed as inhibition of thymol-induced Ca2+ response preincubated for 5 mins followed by...More data for this Ligand-Target Pair
Affinity DataEC50: 4.60E+3nMAssay Description:Agonist activity at rat TRPV3 stably transfected in HEK293 cells assessed as increase in calcium influx in presence of ionomycin by Fluo-4-AM dye bas...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 2(Rat)
University of Naples Federico Ii
Curated by ChEMBL
University of Naples Federico Ii
Curated by ChEMBL
Affinity DataIC50: 2.00E+4nMAssay Description:Antagonist activity at rat TRPV2 expressed in HEK293 cells assessed as inhibition of LPC-induced Ca2+ response preincubated for 5 mins followed by LP...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Human)
University of Naples Federico Ii
Curated by ChEMBL
University of Naples Federico Ii
Curated by ChEMBL
Affinity DataIC50: 2.00E+4nMAssay Description:Antagonist activity at human TRPV1 expressed in HEK293 cells assessed as inhibition of capsaicin-induced Ca2+ response preincubated for 5 mins follow...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1(Human)
University of Naples Federico Ii
Curated by ChEMBL
University of Naples Federico Ii
Curated by ChEMBL
Affinity DataEC50: 4.50E+3nMAssay Description:Agonist activity at human TRPV1 stably transfected in HEK293 cells assessed as increase in calcium influx in presence of ionomycin by Fluo-4-AM dye b...More data for this Ligand-Target Pair