BDBM50542599 CHEMBL4649331

SMILES Cc1cnc2c(c1)-c1ccc(Cl)cc1N(c1ccc(NCCNC3CCOCC3)cc1)C(=O)C2(C)C

InChI Key InChIKey=BMTLFAAUMAGIHF-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50542599   

TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Human)
Daiichi Sankyo

Curated by ChEMBL

LigandBDBM50542599(CHEMBL4649331)Copy SMILESCopy InChI

Affinity DataIC50: 1.60E+3nMAssay Description:Antagonist activity at PTHR1 (unknown origin) expressed in CHOK1 cells co-expressing Gs/Gq assessed as reduction in human PTH (1 to 34 residues)-indu...More data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sidSimilars

In Depth
Date in BDB:
8/13/2021
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