BDBM50541721 CHEMBL4633927

SMILES Cn1cc2n(CCCCF)c(=O)c(C(=O)NC34CC5CC(CC(C5)C3)C4)c(O)c2n1

InChI Key

Data  2 KI  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50541721   

TargetCannabinoid receptor 2(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50541721(CHEMBL4633927)
Affinity DataEC50:  270nMAssay Description:Inverse agonist activity at recombinant human CB2R expressed in CHOK1 cells assessed as increase in NKH477-stimulated intracellular cAMP levels after...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50541721(CHEMBL4633927)
Affinity DataKi:  2.10nMAssay Description:Displacement of [3H]-CP-55,940 from recombinant human CB2R expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50541721(CHEMBL4633927)
Affinity DataKi:  532nMAssay Description:Displacement of [3H]-CP-55,940 from recombinant human CB1R expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed