BDBM50537161 CHEMBL4514739

SMILES Cc4ccc(NC(=O)C[C@H](CCC(=O)[O-])c2noc(c1cc(CC(C)C)on1)c2C3CC3)c(Cl)c4

InChI Key InChIKey=PNYLCKXRNBEDMB-UHFFFAOYSA-M

Data  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50537161   

TargetNuclear receptor ROR-gamma(Human)
Kyoto Prefectural University of Medicine

Curated by ChEMBL
LigandPNGBDBM50537161(CHEMBL4514739)
Affinity DataEC50:  14nMAssay Description:Inhibition of human GAL4-fused RORgamma LBD transcriptional activity expressed in CHOK1 cells after 2 days by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details Article
PubMed