BDBM50534729 CHEMBL4516155

SMILES CN1CCN(C\C=C\C(=O)N2CCCOc3cc4ncnc(Nc5ccc(F)c(Cl)c5)c4cc23)CC1

InChI Key InChIKey=IYPLCHNCAKYCFM-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50534729   

TargetEpidermal growth factor receptor(Human)
Jiangsu Aosaikang Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50534729(CHEMBL4516155)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of EGFR phosphorylation in EGF-stimulated human KB cells preincubated for 1 hr followed by EGF stimulation measured after 6 mins by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2021
Entry Details Article
PubMed