BDBM50532004 CHEMBL4593085

SMILES Cc1cc(NC(=O)Cc2ccc(cc2)-c2ccc(Cl)c(Cl)c2)n(n1)C1CCCCC1

InChI Key InChIKey=QSAGPGILKUZXIU-UHFFFAOYSA-N

Data  2 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50532004   

TargetG protein-activated inward rectifier potassium channel 1(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50532004(CHEMBL4593085)
Affinity DataEC50:  4.47E+3nMAssay Description:Activation of human GIRK1/2 expressed in HEK293 cells co-expressing rat mGlu8 by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetG protein-activated inward rectifier potassium channel 4(Human)
University of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50532004(CHEMBL4593085)
Affinity DataEC50:  4.35E+3nMAssay Description:Activation of human GIRK1/4 expressed in HEK293 cells co-expressing rat mGlu8 by thallium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed