BDBM50531609 CHEMBL4437432

SMILES ONC(=O)c1ccc2C(=O)c3ccccc3C(=O)c2c1

InChI Key InChIKey=CNGWNOQUKFLVKK-UHFFFAOYSA-N

Data  11 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 11 hits for monomerid = 50531609   

TargetHistone deacetylase 3(Human)
Keimyung University

Curated by ChEMBL
LigandPNGBDBM50531609(CHEMBL4437432)
Affinity DataIC50: 3.95E+3nMAssay Description:Inhibition of human recombinant HDAC3 using fluorogenic HDAC substrate-3 by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetHistone deacetylase 6(Human)
Keimyung University

Curated by ChEMBL
LigandPNGBDBM50531609(CHEMBL4437432)
Affinity DataIC50: 56nMAssay Description:Inhibition of human recombinant HDAC6 using fluorogenic HDAC substrate-3 by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetHistone deacetylase 2(Human)
Keimyung University

Curated by ChEMBL
LigandPNGBDBM50531609(CHEMBL4437432)
Affinity DataIC50: 4.62E+3nMAssay Description:Inhibition of HDAC2 (unknown origin) using fluorogenic HDAC substrate-3 by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetHistone deacetylase 8(Human)
Keimyung University

Curated by ChEMBL
LigandPNGBDBM50531609(CHEMBL4437432)
Affinity DataIC50: 599nMAssay Description:Inhibition of human recombinant HDAC8 using fluorogenic HDAC substrate class 2A by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetHistone deacetylase 5(Human)
Keimyung University

Curated by ChEMBL
LigandPNGBDBM50531609(CHEMBL4437432)
Affinity DataIC50: 1.36E+3nMAssay Description:Inhibition of human recombinant HDAC5 using fluorogenic HDAC substrate class 2A by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetHistone deacetylase 7(Human)
Keimyung University

Curated by ChEMBL
LigandPNGBDBM50531609(CHEMBL4437432)
Affinity DataIC50: 1.04E+4nMAssay Description:Inhibition of human recombinant HDAC7 using fluorogenic HDAC substrate class 2A by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetHistone deacetylase 9(Human)
Keimyung University

Curated by ChEMBL
LigandPNGBDBM50531609(CHEMBL4437432)
Affinity DataIC50: 7.78E+3nMAssay Description:Inhibition of human recombinant HDAC9 using fluorogenic HDAC substrate class 2A by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetHistone deacetylase 11(Human)
Keimyung University

Curated by ChEMBL
LigandPNGBDBM50531609(CHEMBL4437432)
Affinity DataIC50: 8.00E+4nMAssay Description:Inhibition of human recombinant HDAC11 using fluorogenic HDAC substrate class 2A by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Keimyung University

Curated by ChEMBL
LigandPNGBDBM50531609(CHEMBL4437432)
Affinity DataIC50: 910nMAssay Description:Inhibition of human recombinant HDAC1 using fluorogenic HDAC substrate-3 by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetHistone deacetylase 4(Human)
Keimyung University

Curated by ChEMBL
LigandPNGBDBM50531609(CHEMBL4437432)
Affinity DataIC50: 5.61E+3nMAssay Description:Inhibition of human recombinant HDAC4 using fluorogenic HDAC substrate class 2A by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetPolyamine deacetylase HDAC10(Human)
Keimyung University

Curated by ChEMBL
LigandPNGBDBM50531609(CHEMBL4437432)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of HDAC10 (unknown origin) by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed