BDBM50526327 CHEMBL4562084::US10752616, Code No. BHBA-023

SMILES Cc1ccc(C)c2oc(nc12)-c1nc(no1)-c1ccc(cc1)C(O)=O

InChI Key InChIKey=VKSMQHIHCUMOQU-UHFFFAOYSA-N

Data  6 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 6 hits for monomerid = 50526327   

TargetRetinoic acid receptor beta(Human)
King''S College London

US Patent
LigandPNGBDBM50526327(CHEMBL4562084 | US10752616, Code No. BHBA-023)
Affinity DataEC50:  11nMAssay Description:Transcriptional transactivation assays were performed with gal4 fusion receptor constructs, created using each of the RAR ligand binding domains of e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/11/2021
Entry Details
Go to US Patent

TargetRetinoic acid receptor alpha(Human)
King''S College London

US Patent
LigandPNGBDBM50526327(CHEMBL4562084 | US10752616, Code No. BHBA-023)
Affinity DataEC50:  114nMAssay Description:Transcriptional transactivation assays were performed with gal4 fusion receptor constructs, created using each of the RAR ligand binding domains of e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/11/2021
Entry Details
Go to US Patent

TargetRetinoic acid receptor gamma(Human)
King''S College London

US Patent
LigandPNGBDBM50526327(CHEMBL4562084 | US10752616, Code No. BHBA-023)
Affinity DataEC50:  83nMAssay Description:Transcriptional transactivation assays were performed with gal4 fusion receptor constructs, created using each of the RAR ligand binding domains of e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/11/2021
Entry Details
Go to US Patent

TargetRetinoic acid receptor beta(Mouse)
King'S College

Curated by ChEMBL
LigandPNGBDBM50526327(CHEMBL4562084 | US10752616, Code No. BHBA-023)
Affinity DataEC50:  11nMAssay Description:Transactivation of GAL4-fused mouse RARbeta-LBD expressed in COS-7 cells after 24 hrs by bright-Glo reagent based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetRetinoic acid receptor alpha(Mouse)
King'S College

Curated by ChEMBL
LigandPNGBDBM50526327(CHEMBL4562084 | US10752616, Code No. BHBA-023)
Affinity DataEC50:  114nMAssay Description:Transactivation of GAL4-fused mouse RARalpha-LBD expressed in COS-7 cells after 24 hrs by bright-Glo reagent based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetRetinoic acid receptor gamma(Mouse)
King'S College

Curated by ChEMBL
LigandPNGBDBM50526327(CHEMBL4562084 | US10752616, Code No. BHBA-023)
Affinity DataEC50:  10nMAssay Description:Transactivation of GAL4-fused mouse RARgamma-LBD expressed in COS-7 cells after 24 hrs by bright-Glo reagent based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed