BDBM50525952 CHEMBL4542977

SMILES CN1CCN(CC1)c1nc2c(F)cccc2c(=O)n1-c1ccc(Cc2ccccc2)cc1

InChI Key InChIKey=HZAQSUDKHPXQSV-UHFFFAOYSA-N

Data  1 EC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50525952   

TargetTransient receptor potential cation channel subfamily V member 4(Human)
Asahi Kasei Medical

Curated by ChEMBL

LigandBDBM50525952(CHEMBL4542977)Copy SMILESCopy InChI

Affinity DataEC50:  670nMAssay Description:Agonist activity at recombinant human TRPV4 expressed in HEK293 cells assessed as increase in intracellular calcium level after 30 mins by Fura-2 AM/...More data for this Ligand-Target Pair

Target InfoPDB
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sidSimilars

In Depth
Date in BDB:
2/25/2021
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